Halogen Bonding Increases the Potency and Isozyme Selectivity of Protein Arginine Deiminase 1 Inhibitors

Author:

Mondal Santanu1,Gong Xuefeng2,Zhang Xiaoqian2,Salinger Ari J.13,Zheng Li1,Sen Sudeshna1,Weerapana Eranthie3,Zhang Xuesen2,Thompson Paul R.1ORCID

Affiliation:

1. Department of Biochemistry and Molecular PharmacologyUniversity of Massachusetts Medical School 364 Plantation street Worcester MA 01605 USA

2. State Key Laboratory of Reproductive MedicineNanjing Medical University Nanjing 211166 China

3. Department of ChemistryBoston College Chestnut Hill MA 02467 USA

Funder

National Institute of General Medical Sciences

Publisher

Wiley

Subject

General Chemistry,Catalysis

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