Synthesis and Biological Evaluation of Phenyl Substituted 1H-1,2,4-Triazoles as Non-Steroidal Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 2
Author:
Publisher
Wiley
Subject
Drug Discovery,Pharmaceutical Science
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1. Inhibitors of 17β-hydroxysteroid dehydrogenase type 1, 2 and 14: Structures, biological activities and future challenges;Molecular and Cellular Endocrinology;2019-06
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3. N-acylimino-substituted 2-oxa-7-azaspiro[4.4]nona-3,6,8-trienes in the synthesis of 3-(1H-1,2,4-triazol-3-yl)-3H-pyrrole-4-carbonitriles;Russian Journal of Organic Chemistry;2017-11
4. Type 2 17-β hydroxysteroid dehydrogenase as a novel target for the treatment of osteoporosis;Future Medicinal Chemistry;2015-08
5. Metabolic stability optimization and metabolite identification of 2,5-thiophene amide 17β-hydroxysteroid dehydrogenase type 2 inhibitors;European Journal of Medicinal Chemistry;2014-11
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