Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain-Barrier-Permeating Compounds

Author:

Van der Poorten Olivier1,Legrand Baptiste2,Vezenkov Lubomir L.2,García-Pindado Júlia3,Bettache Nadir2,Knuhtsen Astrid4,Pedersen Daniel Sejer4,Sánchez-Navarro Macarena3,Martinez Jean2,Teixidó Meritxell3,Garcia Marcel2,Tourwé Dirk1,Amblard Muriel2,Ballet Steven1

Affiliation:

1. Research Group of Organic Chemistry; Departments of Chemistry and Bioengineering Sciences; Vrije Universiteit Brussel; Pleinlaan 2 1050 Brussels Belgium

2. Institut des Biomolécules Max Mousseron (IBMM); UMR 5247; Université de Montpellier; CNRS; ENSCM; 15 Avenue Charles Flahault 34093 Montpellier, Cedex 5 France

3. Institute for Research in Biomedicine (IRB Barcelona); The Barcelona Institute of Science and Technology (BIST); Baldiri Reixac 10 08028 Barcelona Spain

4. Department of Drug Design and Pharmacology; University of Copenhagen; Jagtvej 162 2100 Copenhagen Denmark

Funder

Agentschap voor Innovatie door Wetenschap en Technologie

Carlsberg and Lunbeck Foundation

CNRS

Université de Montpellier

Mineco-feder

Generalitat de Catalunya

Publisher

Wiley

Subject

Organic Chemistry,Molecular Biology,Molecular Medicine,Biochemistry

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