Efforts towards an On‐Target Version of the Groebke–Blackburn–Bienaymé (GBB) Reaction for Discovery of Druglike Urokinase (uPA) Inhibitors-Reference-Cited by-同舟云学术

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Efforts towards an On‐Target Version of the Groebke–Blackburn–Bienaymé (GBB) Reaction for Discovery of Druglike Urokinase (uPA) Inhibitors

Published:2019-08-29 Issue:53 Volume:25 Page:12380-12393
ISSN:0947-6539
Container-title:Chemistry – A European Journal
language:en
Short-container-title:Chem. Eur. J.

Author:

Gladysz Rafaela¹^ORCID,Vrijdag Johannes¹²,Van Rompaey Dries¹,Lambeir Anne‐Marie²,Augustyns Koen¹,De Winter Hans¹,Van der Veken Pieter¹^ORCID

Affiliation:

1. Laboratory of Medicinal Chemistry (UAMC)Department of Pharmaceutical SciencesUniversity of Antwerp Universiteitsplein 1 2610 Wilrijk Belgium

2. Laboratory of Medical BiochemistryDepartment of, Pharmaceutical SciencesUniversity of Antwerp Universiteitsplein 1 2610 Wilrijk Belgium

Publisher

Wiley

Subject

General Chemistry,Catalysis,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/chem.201901917

Reference76 articles.

1. Kinetic target-guided synthesis in drug discovery and chemical biology: a comprehensive facts and figures survey

2. Protein-Templated Fragment Ligations-From Molecular Recognition to Drug Discovery

3. Proteintemplat-gesteuerte Fragmentligationen - von der molekularen Erkennung zur Wirkstofffindung

4. New insights into the kinetic target-guided synthesis of protein ligands

5. Dynamic combinatorial chemistry: a tool to facilitate the identification of inhibitors for protein targets

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4. Linkers in fragment-based drug design: an overview of the literature;Expert Opinion on Drug Discovery;2023-07-19

5. Going beyond Binary: Rapid Identification of Protein–Protein Interaction Modulators Using a Multifragment Kinetic Target-Guided Synthesis Approach;Journal of Medicinal Chemistry;2023-03-31

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