New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition-Reference-Cited by-同舟云学术

New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition

Published:2022-04-15 Issue:7 Volume:355 Page:2200024
ISSN:0365-6233
Container-title:Archiv der Pharmazie
language:en
Short-container-title:Archiv der Pharmazie

Author:

Abdel‐Aziz Salah A.¹²,Taher Ehab S.³,Lan Ping⁴,El‐Koussi Nawal A.²⁵,Salem Ola I. A.⁶,Gomaa Hesham A. M.⁷,Youssif Bahaa G. M.⁶^ORCID

Affiliation:

1. Department of Pharmaceutical Medicinal Chemistry, Faculty of Pharmacy Al‐Azhar University Assiut Egypt

2. Department of Pharmaceutical Chemistry, Faculty of Pharmacy Deraya University Minia Egypt

3. Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy Al‐Azhar University Assiut Egypt

4. Institute for Advanced and Applied Chemical Synthesis Jinan University Guangzhou China

5. Department of Pharmaceutical Medicinal Chemistry, Faculty of Pharmacy Assiut University Assiut Egypt

6. Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy Assiut University Assiut Egypt

7. Pharmacology Department, College of Pharmacy Jouf University Sakaka Saudi Arabia

Publisher

Wiley

Subject

Drug Discovery,Pharmaceutical Science

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/ardp.202200024

Reference56 articles.

1. COX-2 Selective Nonsteroidal Anti-Inflammatory Drugs

2. 1-(4-Methane(amino)sulfonylphenyl)-3-(4-substituted-phenyl)-5-(4-trifluoromethylphenyl)-1H-2-pyrazolines/pyrazoles as potential anti-inflammatory agents

3. Gastrointestinal Damage Associated with the Use of Nonsteroidal Antiinflammatory Drugs

4. Design, synthesis, and biological evaluation of new pyrimidine-5-carbonitrile derivatives bearing 1,3-thiazole moiety as novel anti-inflammatory EGFR inhibitors with cardiac safety profile

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