Synthesis, Anti-Methicillin-resistant S. aureus (MRSA) Evaluation, Quantitative Structure-Activity Relationship and Molecular Modeling Studies of Some Novel Bis-indoles as Prospective MRSA Pyruvate Kinase Inhibitors

Author:

El Sayed Mardia T.1,Sabry Nermien M.1,Hamdy Nehal A.1,Voronkov Andrey2,Ogungbe Ifedayo V.3,Balakin Konstantin4,Abdel-Aziz Mohamed S.5

Affiliation:

1. Applied Organic Chemistry Department, National Research Centre, El Behous street, 12311-Dokki, Egypt

2. Digital Bio Pharm Ltd., 145-157 St. John Street, London, EC1V 4PW, United Kingdom

3. Department of Chemistry & Biochemistry, Jackson State University, 1400 J. R. Lynch Street, P.O. Box 17910-Jackson, MS 39217-0510, United States

4. Moscow Institute of Physic and Technology (State University), Moscow 119991, Russian Federation

5. Microbial Chemistry Department, National Research Centre, El Behous street, 12311-Dokki, Egypt

Publisher

Bentham Science Publishers Ltd.

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

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