Discovery of Selective Estrogen Receptor Covalent Antagonists for the Treatment of ERαWT and ERαMUT Breast Cancer

Author:

Puyang Xiaoling,Furman Craig,Zheng Guo Zhu,Wu Zhenhua J.,Banka Deepti,Aithal Kiran,Agoulnik Sergei,Bolduc David M.,Buonamici Silvia,Caleb Benjamin,Das Subhasree,Eckley Sean,Fekkes Peter,Hao Ming-Hong,Hart Andrew,Houtman RenéORCID,Irwin Sean,Joshi Jaya J.,Karr Craig,Kim Amy,Kumar Namita,Kumar Pavan,Kuznetsov Galina,Lai Weidong G.,Larsen Nicholas,Mackenzie Crystal,Martin Lesley-Ann,Melchers Diana,Moriarty Alyssa,Nguyen Tuong-Vi,Norris John,O'Shea Morgan,Pancholi Sunil,Prajapati Sudeep,Rajagopalan Sujatha,Reynolds Dominic J.,Rimkunas Victoria,Rioux Nathalie,Ribas Ricardo,Siu Amy,Sivakumar Sasirekha,Subramanian Vanitha,Thomas Michael,Vaillancourt Frédéric H.,Wang John,Wardell Suzanne,Wick Michael J.,Yao Shihua,Yu Lihua,Warmuth Markus,Smith Peter G.,Zhu Ping,Korpal Manav

Funder

Breast Cancer Now Toby Robins Research Centre

Publisher

American Association for Cancer Research (AACR)

Subject

Oncology

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