Prediction of a potentially effective dose in humans for BAY 60-5521, a potent inhibitor of cholesteryl ester transfer protein (CETP) by allometric species scaling and combined pharmacodynamic and physiologically-based pharmacokinetic modelling-Reference-Cited by-同舟云学术

Prediction of a potentially effective dose in humans for BAY 60-5521, a potent inhibitor of cholesteryl ester transfer protein (CETP) by allometric species scaling and combined pharmacodynamic and physiologically-based pharmacokinetic modelling

Published:2012-01-06 Issue:2 Volume:73 Page:219-231
ISSN:0306-5251
Container-title:British Journal of Clinical Pharmacology
language:en
Short-container-title:

Author:

Weber Olaf,Willmann Stefan,Bischoff Hilmar,Li Volkhart,Vakalopoulos Alexandros,Lustig Klemens,Hafner Frank-Thorsten,Heinig Roland,Schmeck Carsten,Buehner Klaus

Publisher

Wiley

Subject

Pharmacology (medical),Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1365-2125.2011.04064.x/fullpdf

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4. Prediction of hepatic metabolic clearance based on interspecies allometric scaling techniques and in vitro-in vivo correlations;Lave;Clin Pharmacokinetet,1999

5. Comparison of the disposition of two novel combined thromboxane synthase inhibitors/thromboxane A2 receptor antagonists in the isolated perfused rat liver;Gardner;Xenobiotica,1995

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