Novel µ opioid antagonists derived from the µ opioid agonists endomorphin and [Dmt 1 ]DALDA (H‐Dmt‐D‐Arg‐Phe‐Lys‐NH 2 )-Reference-Cited by-同舟云学术

Novel µ opioid antagonists derived from the µ opioid agonists endomorphin and [Dmt 1 ]DALDA (H‐Dmt‐D‐Arg‐Phe‐Lys‐NH 2 )

Published:2020-08-02 Issue:5 Volume:96 Page:1305-1314
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Shi Saijian¹,Xu Jian¹,Feng LingLing¹,Fan Xin¹,Chen Zhen¹,Qin Yajuan¹,Chung Nga N.²^ORCID,Li Tingyou¹³,Schiller Peter W.²⁴^ORCID

Affiliation:

1. School of Pharmacy Nanjing Medical University Nanjing China

2. Laboratory of Chemical Biology and Peptide Research Montreal Clinical Research Institute Montreal QC Canada

3. Key Laboratory of Targeted Intervention of Cardiovascular Disease Collaborative Innovation Center for Cardiovascular Disease Translational Medicine Nanjing Medical University Nanjing China

4. Department of Pharmacology and Physiology Université de Montréal Montreal QC Canada

Funder

Canadian Institutes of Health Research

National Institutes of Health

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/cbdd.13743

Reference28 articles.

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5. Synthesis and pharmacological characterization in vitro of cyclic enkephalin analogs: effect of conformational constraints on opiate receptor selectivity

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