In vitro and in vivo characterization of the bifunctional μ and δ opioid receptor ligand UFP‐505-Reference-Cited by-同舟云学术

In vitro and in vivo characterization of the bifunctional μ and δ opioid receptor ligand UFP‐505

Published:2018-05-14 Issue:14 Volume:175 Page:2881-2896
ISSN:0007-1188
Container-title:British Journal of Pharmacology
language:en
Short-container-title:British Journal of Pharmacology

Author:

Dietis N¹^ORCID,Niwa H¹,Tose R¹,McDonald J¹,Ruggieri V²,Filaferro M³,Vitale G⁴,Micheli L⁵,Ghelardini C⁵,Salvadori S⁶,Calo G⁶^ORCID,Guerrini R⁷,Rowbotham D J⁸,Lambert D G¹^ORCID

Affiliation:

1. Department of Cardiovascular SciencesUniversity of Leicester, Division of Anaesthesia, Critical Care and Pain Management, Leicester Royal Infirmary Leicester UK

2. Department of Oncology Haematology and Respiratory DiseasesUniversity of Modena and Reggio Emilia Modena Italy

3. Department of Biomedical, Metabolic and Neuro‐SciencesUniversity of Modena and Reggio Emilia Modena Italy

4. Section of Pharmacology, Department of Life SciencesUniversity of Modena and Reggio Emilia Modena Italy

5. Department of Preclinical and Clinical PharmacologyUniversity of Florence Florence Italy

6. Department of Experimental and Clinical Medicine, Section of PharmacologyUniversity of Ferrara Ferrara Italy

7. Department of Pharmaceutical SciencesUniversity of Ferrara Ferrara Italy

8. Department of Health SciencesUniversity of Leicester, Division of Anaesthesia, Critical Care and Pain Management, Leicester Royal Infirmary Leicester UK

Funder

HOPE Against Cancer

Publisher

Wiley

Subject

Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/bph.14199

Reference63 articles.

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4. Relative Opioid Efficacy Is Determined by the Complements of the G Protein-Coupled Receptor Desensitization Machinery

5. G Protein independent phosphorylation and internalization of the δ-opioid receptor

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