Ribociclib shows potential for pharmacokinetic drug-drug interactions being a substrate of ABCB1 and potent inhibitor of ABCB1, ABCG2 and CYP450 isoforms in vitro-Reference-Cited by-同舟云学术

Ribociclib shows potential for pharmacokinetic drug-drug interactions being a substrate of ABCB1 and potent inhibitor of ABCB1, ABCG2 and CYP450 isoforms in vitro

Published:2018-08 Issue: Volume:154 Page:10-17
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Sorf Ales,Hofman Jakub,Kučera Radim,Staud Frantisek,Ceckova Martina

Funder

Czech Science Foundation

Charles University

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

Reference39 articles.

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4. Spectrum and degree of CDK drug interactions predicts clinical performance;Chen;Mol. Cancer Ther.,2016

5. Chemoproteomics reveals novel protein and lipid kinase targets of clinical CDK4/6 inhibitors in lung cancer;Sumi;ACS Chem. Biol.,2015

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