Receptor antagonism/agonism can be uncoupled from pharmacoperone activity

Author:

Janovick Jo Ann,Spicer Timothy P.,Smith Emery,Bannister Thomas D.,Kenakin Terry,Scampavia Louis,Conn P. MichaelORCID

Funder

National Institutes of Health

Publisher

Elsevier BV

Subject

Endocrinology,Molecular Biology,Biochemistry

Reference36 articles.

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4. Pharmacoperones and the calcium sensing receptor: exogenous and endogenous regulators;Breitwieser;Pharmacol. Res. Off. J. Ital. Pharmacol. Soc.,2014

5. Behind the curtain: cellular mechanisms for allosteric modulation of calcium-sensing receptors;Cavanaugh;Br. J. Pharmacol.,2012

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