Receptor antagonism/agonism can be uncoupled from pharmacoperone activity
Author:
Funder
National Institutes of Health
Publisher
Elsevier BV
Subject
Endocrinology,Molecular Biology,Biochemistry
Reference36 articles.
1. Properties of a new radioiodinated antagonist for human vasopressin V2 and V1a receptors;Ala;Eur. J. Pharmacol.,1997
2. Interplay between two allosteric sites and their influence on agonist binding in human mu opioid receptor;Bartuzi;J. Chem. Inf. Model,2016
3. The calcium sensing receptor life cycle: trafficking, cell surface expression, and degradation;Breitwieser;Best. Pract. Res. Clin. Endocrinol. Metab.,2013
4. Pharmacoperones and the calcium sensing receptor: exogenous and endogenous regulators;Breitwieser;Pharmacol. Res. Off. J. Ital. Pharmacol. Soc.,2014
5. Behind the curtain: cellular mechanisms for allosteric modulation of calcium-sensing receptors;Cavanaugh;Br. J. Pharmacol.,2012
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