Discovery of cycloalkyl-fused N -thiazol-2-yl-benzamides as tissue non-specific glucokinase activators: Design, synthesis, and biological evaluation-Reference-Cited by-同舟云学术

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Discovery of cycloalkyl-fused N -thiazol-2-yl-benzamides as tissue non-specific glucokinase activators: Design, synthesis, and biological evaluation

Published:2017-10 Issue: Volume:139 Page:128-152
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Wang Zhengyu,Shi Xiaofan,Zhang Huan,Yu Liang,Cheng Yanhua,Zhang Hefeng,Zhang Huibin,Zhou Jinpei,Chen Jing,Shen Xu,Duan Wenhu

Funder

Personalized Medicines--Molecular Signature-based Drug Discovery and Development

Strategic Priority Research Program of the Chinese Academy of Sciences

Institutes for Drug Discovery and Development

Chinese Academy of Sciences

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference57 articles.

1. Management of type 2 diabetes: new and future developments in treatment;Tahrani;Lancet,2011

2. The diabetes pandemic;Lancet,2011

3. Lessons from glucokinase activators: the problem of declining efficacy;Agius;Expert Opin. Ther. Pat.,2014

4. Assessing the potential of glucokinase activators in diabetes therapy;Matschinsky;Nat. Rev. Drug Discov.,2009

5. Strategies for the design of hepatoselective glucokinase activators to treat type 2 diabetes;Pfefferkorn;Expert Opin. Drug Discov.,2013

Cited by 11 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Molecular docking, 2D-QSAR and ADMET studies of 4-sulfonyl-2-pyridone heterocycle as a potential glucokinase activator;Results in Chemistry;2023-12

2. Identification of small-molecule glucokinase activator for type-2-diabetes treatment: a structure-based virtual screening approach;Molecular Simulation;2023-09-14

3. Conformational, Reactivity Analysis, Wavefunction-Based Properties, Molecular Docking and Simulations of a Benzamide Derivative with Potential Antitumor Activity-DFT and MD Simulations;Polycyclic Aromatic Compounds;2022-02-16

4. A comprehensive review on glucokinase activators: Promising agents for the treatment of Type 2 diabetes;Chemical Biology & Drug Design;2021-11-10

5. Design and synthesis of newer N-benzimidazol-2yl benzamide analogues as allosteric activators of human glucokinase;Medicinal Chemistry Research;2021-01-13

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