Identification of fused 16β,17β-oxazinone-estradiol derivatives as a new family of non-estrogenic 17β-hydroxysteroid dehydrogenase type 1 inhibitors-Reference-Cited by-同舟云学术

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Identification of fused 16β,17β-oxazinone-estradiol derivatives as a new family of non-estrogenic 17β-hydroxysteroid dehydrogenase type 1 inhibitors

Published:2015-03 Issue: Volume:93 Page:470-480
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Maltais René,Trottier Alexandre,Delhomme Audrey,Barbeau Xavier,Lagüe Patrick,Poirier Donald

Funder

Canadian Institutes of Health Research

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference36 articles.

1. Integrated view on 17beta-hydroxysteroid dehydrogenase;Moeller;Mol. Cell. Endocrinol.,2009

2. 17beta-hydroxysteroid dehydrogenase: inhibitors and inhibitor design;Penning;Endocr. Relat. Cancer,1996

3. The estrogen receptor as a target for rational drug design;von Angerer,1995

4. Full oestrogenic activity of C19-delta 5 adrenal steroids in rat pituitary lactotrophs and somatotrophs;Simard;Mol. Cell. Endocrinol.,1988

5. 17β-Hydroxysteroid dehydrogenases in human breast cancer;Nagasaki;Ann. N. Y. Acad. Sci.,2009

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2. RuPHOX-Ru-Catalyzed Selective Asymmetric Hydrogenation of Exocyclic α,β-Unsaturated Pentanones;Organometallics;2019-08-07

3. Inhibitors of 17β-hydroxysteroid dehydrogenase type 1, 2 and 14: Structures, biological activities and future challenges;Molecular and Cellular Endocrinology;2019-06

4. Steroidal Anticancer Agents: An Overview of Estradiol-related Compounds;Anti-Cancer Agents in Medicinal Chemistry;2018-08-21

5. Synthesis of novel 16-E-(arylidene)-3-methoxy-α-estrones via a palladium catalysed Suzuki-Miyaura reaction;Tetrahedron Letters;2018-01

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