A road map for prioritizing warheads for cysteine targeting covalent inhibitors-Reference-Cited by-同舟云学术

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A road map for prioritizing warheads for cysteine targeting covalent inhibitors

Published:2018-12 Issue: Volume:160 Page:94-107
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Ábrányi-Balogh Péter,Petri László,Imre Tímea,Szijj Péter,Scarpino Andrea,Hrast Martina^ORCID,Mitrović Ana,Fonovič Urša Pečar,Németh Krisztina,Barreteau Hélène,Roper David I.,Horváti Kata^ORCID,Ferenczy György G.,Kos Janko,Ilaš Janez^ORCID,Gobec Stanislav^ORCID,Keserű György M.^ORCID

Funder

National Brain Research Program

MSCA ETN FRAGNET

Hungarian Science Foundation OTKA

Hungarian Academy of Sciences postdoctoral fellowship

Slovenian Research Agency

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference57 articles.

1. Targeted covalent inhibitors for drug design;Baillie;Angew. Chem. Int. Ed. Engl. Transl,2016

2. Covalent protein modification: the current landscape of residue-specific electrophiles;Shannon;Curr. Opin. Chem. Biol.,2015

3. Relationship Between the Occurrence of Cysteine in Proteins and the Complexity of Organisms;Miseta;Mol. Biol. Evol.,2000

4. Targeting non-catalytic cysteine residues through structure-guided drug discovery;Hallenbeck;Curr. Top. Med. Chem.,2017

5. Progress with covalent small-molecule kinase inhibitors;Zhao;Drug Discov. Today,2018

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2. Quantum Chemical Characterization of Rotamerism in Thio-Michael Additions for Targeted Covalent Inhibitors;Journal of Chemical Information and Modeling;2024-09-12

3. Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads;Communications Chemistry;2024-09-09

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5. Contribution of Noncovalent Recognition and Reactivity to the Optimization of Covalent Inhibitors: A Case Study on KRas^G12C;ACS Chemical Biology;2024-07-11

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