Synthesis and biological evaluation of a novel sigma-1 receptor antagonist based on 3,4-dihydro-2(1H)-quinolinone scaffold as a potential analgesic-Reference-Cited by-同舟云学术

Synthesis and biological evaluation of a novel sigma-1 receptor antagonist based on 3,4-dihydro-2(1H)-quinolinone scaffold as a potential analgesic

Published:2014-05 Issue: Volume:79 Page:216-230
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Lan Yu,Chen Yin,Xu Xiangqing,Qiu Yinli,Liu Shicheng,Liu Xin,Liu Bi-Feng,Zhang Guisen

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference48 articles.

1. Pain management: a fundamental human right;Brennan;Anesthesia & Analgesia,2007

2. Treatment of the chronic non-cancer pain;Turk;Lancet,2011

3. Further studies on arylpiperazinyl alkyl pyridazinones: discovery of an exceptionally potent, orally active, antinociceptive agent in thermally induced pain;Biancalani;Journal of Medicinal Chemistry,2009

4. γ-aminobutyric acid amides of nortriptyline and fluoxetine display improved pain suppressing activity;Rephaeli;Journal of Medicinal Chemistry,2009

5. The effects of morphine- and nalorphine-like drugs in the nondependent and morphine-dependent chronic spinal dog;Martin;Journal of Pharmacology and Experimental Therapeutics,1976

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