Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability

Author:

Federico Stefano,Khan Tuhina,Fontana Anna,Brogi Simone,Benedetti Rosaria,Sarno Federica,Carullo Gabriele,Pezzotta Alex,Saraswati Akella Prasanth,Passaro Eugenia,Pozzetti Luca,Papa Alessandro,Relitti Nicola,Gemma Sandra,Butini Stefania,Pistocchi Anna,Ramunno Anna,Vincenzi Fabrizio,Varani Katia,Tatangelo Vanessa,Patrussi Laura,Baldari Cosima T.,Saponara Simona,Gorelli Beatrice,Lamponi Stefania,Valoti Massimo,Saccoccia Fulvio,Giannaccari Marialaura,Ruberti Giovina,Herp Daniel,Jung Manfred,Altucci Lucia,Campiani Giuseppe

Funder

MIUR

Campania Region

Associazione Italiana per la Ricerca sul Cancro

Tuscany Region

Airc Italian Foundation for Cancer Research

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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