Design and synthesis of proteolysis targeting chimeras (PROTACs) as an EGFR degrader based on CO-1686
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference38 articles.
1. EGFR mutations and lung cancer;Da;Annu. Rev. Pathol.,2011
2. The biology and management of non-small cell lung cancer;Herbst;Nature,2018
3. Small molecule inhibitors targeting the EGFR/ErbB family of protein-tyrosine kinases in human cancers;Roskoski;Pharmacol. Res.,2019
4. The next tier of EGFR resistance mutations in lung cancer;Tumbrink;Oncogene,2021
5. EGFR mutation and resistance of non-small-cell lung cancer to gefitinib;Kobayashi;N. Engl. J. Med.,2005
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