Inhibitor versus chaperone behaviour of d-fagomine, DAB and LAB sp2-iminosugar conjugates against glycosidases: A structure–activity relationship study in Gaucher fibroblasts-Reference-Cited by-同舟云学术

Inhibitor versus chaperone behaviour of d-fagomine, DAB and LAB sp2-iminosugar conjugates against glycosidases: A structure–activity relationship study in Gaucher fibroblasts

Published:2016-10 Issue: Volume:121 Page:880-891
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Mena-Barragán Teresa,García-Moreno M. Isabel,Nanba Eiji,Higaki Katsumi,Concia Alda Lisa,Clapés Pere,García Fernández José Manuel,Ortiz Mellet Carmen

Funder

JSPS KAKENHI

Takeda Science Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference64 articles.

1. Iminosugars past, present and future: medicines for tomorrow

2. d-Fagomine lowers postprandial blood glucose and modulates bacterial adhesion

3. Sugar-mimic glycosidase inhibitors: natural occurrence, biological activity and prospects for therapeutic application

4. The l-enantiomers of d-sugar-mimicking iminosugars are noncompetitive inhibitors of d-glycohydrolase?

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