Serendipitous discovery of Class I HDAC inhibitors from rational design of molecular glue degraders targeting HDAC-Reference-Cited by-同舟云学术

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Serendipitous discovery of Class I HDAC inhibitors from rational design of molecular glue degraders targeting HDAC

Published:2024-01 Issue: Volume:263 Page:115926
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Chen Di,Lin Shuxian,Zeng Ziwei,An Jianxiong,Yan Wanli,Gu Zhicheng,Chen Lei,He Bin

Funder

National Natural Science Foundation of China

Guizhou Provincial Science and Technology Department

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference34 articles.

1. Synthesis and biological study of class I selective HDAC inhibitors with NO releasing activity;Liu;Bioorg. Chem.,2020

2. Chidamide (CS055/HBI-8000): a new histone deacetylase inhibitor of the benzamide class with antitumor activity and the ability to enhance immune cell-mediated tumor cell cytotoxicity;Ning;Cancer Chemother. Pharmacol.,2012

3. Discovery of novel hit compounds as potential HDAC1 inhibitors: the case of ligand-and structure-based virtual screening;Sirous;Comput. Biol. Med.,2021

4. Design, synthesis and biological evaluation of novel isoindolinone derivatives as potent histone deacetylase inhibitors;Chen;Eur. J. Med. Chem.,2019

5. Design, synthesis and biological evaluation of quinoline derivatives as HDAC class I inhibitors;Chen;Eur. J. Med. Chem.,2017

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