Measurement of total and unbound bictegravir concentrations in plasma and cerebrospinal fluid by UHPLC-MS/MS

Author:

Rigo-Bonnin Raúl,Tiraboschi Juan Manuel,Álvarez-Álvarez Marta,Pérez-Fernández Gloria Ainara,Sanjuás-Iglesias Mercedes,Scévola Sofía,Niubó Jordi,Videla Sebastián,Podzamczer Daniel

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Spectroscopy,Drug Discovery,Pharmaceutical Science,Analytical Chemistry

Reference20 articles.

1. Initial antiretroviral therapy in an integrase inhibitor era: can we do better?;Kelly;Infect. Dis. Clin. North. Am.,2019

2. Bictegravir;Spagnuolo;Curr. Opin. HIV AIDS.,2018

3. Antiviral activity of bictegravir (GS-9883), a novel potent HIV-1 integrase strand transfer inhibitor with an improved resistance profile;Tsiang;Antimicrob. Agents Chemother.,2016

4. Co-formulated bictegravir, emtricitabine, and tenofovir alafenamide versus dolutegravir with emtricitabine and tenofovir alafenamide for initial treatment of HIV-1 infection: week 96 results from a randomised, double-blind, multicentre, phase 3, non-inferiority trial

5. Bictegravir/Emtricitabine/Tenofovir Alafenamide: A review in HIV-1 infection;Deeks;Drugs.,2018

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