A mild and efficient approach to the 6H-oxazolo[3,2-f]pyrimidine-5,7-dione scaffold via unexpected rearrangement of 2,3-dihydropyrimido[6,1-b][1,5,3]dioxazepine-7,9(5H,8H)-diones: synthesis, crystallographic studies, and cytotoxic activity screening-Reference-Cited by-同舟云学术

A mild and efficient approach to the 6H-oxazolo[3,2-f]pyrimidine-5,7-dione scaffold via unexpected rearrangement of 2,3-dihydropyrimido[6,1-b][1,5,3]dioxazepine-7,9(5H,8H)-diones: synthesis, crystallographic studies, and cytotoxic activity screening

Published:2016-02 Issue:7 Volume:57 Page:743-746
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Mieczkowski Adam,Bazlekowa Milena,Bagiński Maciej,Wójcik Jacek,Winczura Alicja,Miazga Agnieszka,Shahmoradi Ghahe Somayeh,Gajda Roman,Woźniak Krzysztof,Tudek Barbara

Funder

Polish Ministry of Science and Higher Education

Centre for Preclinical Research and Technology

European Regional Development Fund and Innovative Economy

National Cohesion Strategy of Poland

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference17 articles.

1. Dyer, R. D.; Harter, W. G.; Hicks, J. L.; Johnson, A. R.; Li, J. J.; Roark, W. H.; Shuler, K. R. WO 02/064599 A1, 2002.

2. Efficient synthesis of bicyclic oxazolino- and thiazolino[3,2-c]pyrimidine-5,7-diones and its application to the synthesis of GnRH antagonists