Discovery and Development of TMPRSS6 Inhibitors Modulating Hepcidin Levels in Human Hepatocytes-Reference-Cited by-同舟云学术

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Discovery and Development of TMPRSS6 Inhibitors Modulating Hepcidin Levels in Human Hepatocytes

Published:2019-11 Issue:11 Volume:26 Page:1559-1572.e9
ISSN:2451-9456
Container-title:Cell Chemical Biology
language:en
Short-container-title:Cell Chemical Biology

Author:

Béliveau François,Tarkar Aarti,Dion Sébastien P.,Désilets Antoine,Ghinet Mariana Gabriela,Boudreault Pierre-Luc,St-Georges Catherine,Marsault Éric,Paone Daniel,Collins Jon,Macphee Colin H.,Campobasso Nino,Groy Arthur,Cottom Josh,Ouellette Michael,Pope Andrew J.,Leduc Richard

Funder

Canadian Institutes of Health Research

Discovery Partnerships with Academia

GlaxoSmithKline

GSK

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,Biochemistry

Reference63 articles.

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2. PHENIX: a comprehensive Python-based system for macromolecular structure solution;Adams;Acta Crystallogr. D Biol. Crystallogr.,2010

3. Membrane-anchored serine proteases in health and disease;Antalis;Prog. Mol. Biol. Transl. Sci.,2011

4. From haystack to needle: finding value with DNA encoded library technology at GSK;Arico-Muendel;MedChemComm,2016

5. Structure-function analysis of ferroportin defines the binding site and an alternative mechanism of action of hepcidin;Aschemeyer;Blood,2018

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1. TMPRSS6 cleaves KCNE1 and causes arrhythmias in iron overload disease;2024-09-10

2. Development of ketobenzothiazole-based peptidomimetic TMPRSS13 inhibitors with low nanomolar potency;2024-08-29

3. Rational In Silico Design of Selective TMPRSS6 Peptidomimetic Inhibitors via Exploitation of the S2 Subpocket;Journal of Medicinal Chemistry;2024-07-19

4. Pre-Infection Innate Immunity Attenuates SARS-CoV-2 Infection and Viral Load in iPSC-Derived Alveolar Epithelial Type 2 Cells;Cells;2024-02-21

5. Pharmacophore-based computational study on inhibitor of TMPRSS6 as hepcidin modulator in an iron overload of beta-thalassaemia;Molecular Simulation;2024-01-17

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