The synthesis of novel GABA uptake inhibitors. Part 2. Synthesis of 5-hydroxytiagabine, a human metabolite of the GABA reuptake inhibitor tiagabine-Reference-Cited by-同舟云学术

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The synthesis of novel GABA uptake inhibitors. Part 2. Synthesis of 5-hydroxytiagabine, a human metabolite of the GABA reuptake inhibitor tiagabine

Published:1994-01 Issue:29 Volume:50 Page:8699-8710
ISSN:0040-4020
Container-title:Tetrahedron
language:en
Short-container-title:Tetrahedron

Author:

Andersen Knud E.,Begtrup Mikael,Chorghade Mukund S.,Lee Elaine C.,Lau Jesper,Lundt Behrend F.,Petersen Hans,Sørensen Per O.,Thøgersen Henning

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference24 articles.

1. The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (Tiagabine) as an anticonvulsant drug candidate

2. Memory failure in epilepsy: retrospective reports and prospective recordings

3. Acid-catalyzed brominations, deuterations, rearrangements, and debrominations of thiophenes under mild conditions

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2. Synthesis and biological evaluation of novel N-substituted nipecotic acid derivatives with an alkyne spacer as GABA uptake inhibitors;Bioorganic & Medicinal Chemistry;2018-07

3. Thiophene-Based Quinomethane Analogs;Advances in Heterocyclic Chemistry;2017

4. Delivering toxicity tests;Chemistry & Industry;2014-10

5. Synthesis and evaluation of N-substituted nipecotic acid derivatives with an unsymmetrical bis-aromatic residue attached to a vinyl ether spacer as potential GABA uptake inhibitors;Bioorganic & Medicinal Chemistry;2013-06

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