Evaluation of carbon-11 labeled 5-(1-methyl-1H-pyrazol-4-yl)-N-(2-methyl-5-(3-(trifluoromethyl)benzamido)phenyl)nicotinamide as PET tracer for imaging of CSF-1R expression in the brain-Reference-Cited by-同舟云学术

Evaluation of carbon-11 labeled 5-(1-methyl-1H-pyrazol-4-yl)-N-(2-methyl-5-(3-(trifluoromethyl)benzamido)phenyl)nicotinamide as PET tracer for imaging of CSF-1R expression in the brain

Published:2021-07 Issue: Volume:42 Page:116245
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

van der Wildt Berend,Nezam Madina,Kooijman Esther J.M.,Reyes Samantha T.,Shen Bin,Windhorst Albert D.,Chin Frederick T.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference37 articles.

1. Expression of the receptor for macrophage colony stimulating factor by brain microglia and its upregulation in brains of patients with Alzheimer’s disease and amyotrophic lateral sclerosis;Akiyama;Brain Res,1994

2. Emerging roles for CSF-1 receptor and its ligands in the nervous system;Chitu;Trends Neurosci,2016

3. Microglia and macrophages in brain homeostasis and disease;Li;Nat Rev Immunol,2018

4. CSF-1R inhibition alters macrophage polarization and blocks glioma progression;Pyonteck;Nat Med,2013

5. Colony-stimulating factor 1 receptor signaling is necessary for microglia viability, unmasking a microglia progenitor cell in the adult brain;Elmore;Neuron,2014

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