Discovery and structure–activity relationship studies of N6-benzoyladenine derivatives as novel BRD4 inhibitors-Reference-Cited by-同舟云学术

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Discovery and structure–activity relationship studies of N6-benzoyladenine derivatives as novel BRD4 inhibitors

Published:2015-03 Issue:5 Volume:23 Page:953-959
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Noguchi-Yachide Tomomi,Sakai Taki,Hashimoto Yuichi,Yamaguchi Takao

Funder

Ministry of Education, Culture, Sports, Science and Technology, Japan

The Japan Society for the Promotion of Science

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference34 articles.

1. Targeting bromodomains: epigenetic readers of lysine acetylation

2. Histone Recognition and Large-Scale Structural Analysis of the Human Bromodomain Family

3. Brd4 Coactivates Transcriptional Activation of NF-κB via Specific Binding to Acetylated RelA

4. Suppression of inflammation by a synthetic histone mimic

5. Brd4 Recruits P-TEFb to Chromosomes at Late Mitosis To Promote G 1 Gene Expression and Cell Cycle Progression

Cited by 22 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Dual inhibitors of HDAC and other epigenetic regulators: A novel strategy for cancer treatment;European Journal of Medicinal Chemistry;2024-01

2. Hybrid Histone Deacetylase Inhibitor: An Effective Strategy for Cancer Therapy;Current Medicinal Chemistry;2023-06

3. Cytotoxic and antitumoral activity of N-(9H-purin-6-yl) benzamide derivatives and related water-soluble prodrugs;Current Molecular Pharmacology;2021-10-14

4. Dual‐target inhibitors of bromodomain and extra‐terminal proteins in cancer: A review from medicinal chemistry perspectives;Medicinal Research Reviews;2021-10-11

5. Cell-surface SLC nucleoside transporters and purine levels modulate BRD4-dependent chromatin states;Nature Metabolism;2021-05

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