Design, synthesis, structural optimization, SAR, in silico prediction of physicochemical properties and pharmacological evaluation of novel & potent thiazolo[4,5-d]pyrimidine corticotropin releasing factor (CRF) receptor antagonists-Reference-Cited by-同舟云学术

Design, synthesis, structural optimization, SAR, in silico prediction of physicochemical properties and pharmacological evaluation of novel & potent thiazolo[4,5-d]pyrimidine corticotropin releasing factor (CRF) receptor antagonists

Published:2022-02 Issue: Volume:169 Page:106084
ISSN:0928-0987
Container-title:European Journal of Pharmaceutical Sciences
language:en
Short-container-title:European Journal of Pharmaceutical Sciences

Author:

Islam Md Rabiul,Teleb Mohamed,Karageorgos Vlasios,Sakellaris Stelios,Papadopoulos Minas,Pirmettis Ioannis,Fronczek Frank R.,Liapakis George,Fahmy Hesham

Publisher

Elsevier BV

Subject

Pharmaceutical Science

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4. Beck, J., Thiazolo[4,5-d]pyrimidines and Pyridines as Corticotropin Releasing Factor (CRF) Antagonist. US Patent, US6107294A,1999: USA; WO-9951608-A1, 1999.

5. Thiazolo[4,5-d]pyrimidine thiones and -ones as corticotropin-releasing hormone (CRH-R1) receptor antagonists;Beck;Bioorg. Med. Chem. Lett.,1999

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