Inhibition of Kv1.3 channels by H-89 (N-[2- (p-bromocinnamylamino)ethyl]-5-isoquinolinesulfonamide) independent of protein kinase A11Abbreviations: AMP-PNP, 5′-adenylyl-imidodiphosphate; CHO, Chinese hamster ovary; H-89, N-[2-(p-bromocinnamylamino)ethyl]-5-isoquinolinesulfonamide; PKA, protein kinase A; PKC, protein kinase C; PKI 5-24, protein kinase A inhibitor 5-24; Rp-cAMPS, adenosine 3′, 5′-cyclic phosphorothioate-Rp-Reference-Cited by-同舟云学术

Inhibition of Kv1.3 channels by H-89 (N-[2- (p-bromocinnamylamino)ethyl]-5-isoquinolinesulfonamide) independent of protein kinase A11Abbreviations: AMP-PNP, 5′-adenylyl-imidodiphosphate; CHO, Chinese hamster ovary; H-89, N-[2-(p-bromocinnamylamino)ethyl]-5-isoquinolinesulfonamide; PKA, protein kinase A; PKC, protein kinase C; PKI 5-24, protein kinase A inhibitor 5-24; Rp-cAMPS, adenosine 3′, 5′-cyclic phosphorothioate-Rp

Published:2001-04 Issue:8 Volume:61 Page:1029-1032
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Choi Jin-Sung,Choi Bok Hee,Hahn Sang June,Yoon Shin Hee,Min Do Sik,Jo Yang-Hyeok,Kim Myung-Suk

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

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4. Effects of the protein kinase A inhibitor H-89 on Ca2+ regulation in isolated ferret ventricular myocytes;Hussain;Pflügers Arch,1999

5. Lo CF, Breitwieser GE. Protein kinase-independent inhibition of muscarinic K+ channels by staurosporine. Am J Physiol 1994;266:C1128–32.

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