Utilization of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold in the design of potent inhibitors of serine proteases: SAR studies using carboxylates-Reference-Cited by-同舟云学术

Utilization of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold in the design of potent inhibitors of serine proteases: SAR studies using carboxylates

Published:2000-05 Issue:5 Volume:8 Page:1005-1016
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Kuang Rongze,Epp Jeffrey B.,Ruan Sumei,Chong Lee S.,Venkataraman Radhika,Tu Juan,He Shu,Truong Tien M.,Groutas William C.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference44 articles.

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3. (c) Hiemstra, P. S.; van Wetering, S.; Stolk, J. Eur. Respir. J. 1998, 12, 1200.

4. The Role of Proteolytic Enzymes in the Development of Pulmonary Emphysema and Periodontal Disease

5. (a) Wiedow, O.; Wiese, F.; Christophers, E. Arch. Dermatol. Res. 1995, 287, 632.

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