Discovery of potent and selective bicyclic A2B adenosine receptor antagonists via bioisosteric amide replacement-Reference-Cited by-同舟云学术

Discovery of potent and selective bicyclic A2B adenosine receptor antagonists via bioisosteric amide replacement

Published:2010-03 Issue:5 Volume:20 Page:1634-1637
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Eastwood Paul,Gonzalez Jacob,Paredes Sergio,Fonquerna Silvia,Cardús Arantxa,Alonso Juan Antonio,Nueda Arsenio,Domenech Teresa,Reinoso Raquel F.,Vidal Bernat

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference26 articles.

1. Adenosine A2b receptors evoke interleukin-8 secretion in human mast cells. An enprofylline-sensitive mechanism with implications for asthma.

2. New insights into the regulation of inflammation by adenosine

3. Differential Expression of Adenosine Receptors in Human Endothelial Cells

4. Mast Cell–Mediated Stimulation of Angiogenesis

5. Hypoxia Modulates Adenosine Receptors in Human Endothelial and Smooth Muscle Cells Toward an A2BAngiogenic Phenotype

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