Discovery of novel N-hydroxy-2-arylisoindoline-4-carboxamides as potent and selective inhibitors of HDAC11-Reference-Cited by-同舟云学术

Discovery of novel N-hydroxy-2-arylisoindoline-4-carboxamides as potent and selective inhibitors of HDAC11

Published:2018-07 Issue:12 Volume:28 Page:2143-2147
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Martin Matthew W.,Lee Jennifer Y.,Lancia David R.,Ng Pui Yee,Han Bingsong,Thomason Jennifer R.,Lynes Maureen S.,Marshall C. Gary,Conti Chiara,Collis Alan,Morales Monica Alvarez,Doshi Kshama,Rudnitskaya Aleksandra,Yao Lili,Zheng Xiaozhang

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference14 articles.

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3. Towards selective inhibition of histone deacetylase isoforms: what has been achieved, where we are and what will be next;Thaler;ChemMedChem,2014

4. Cloning and functional characterization of HDAC11, a novel member of the human histone deacetylase family;Gao;J Biol Chem,2002

5. T-cells lacking HDAC11 have increased effector functions and mediate enhanced alloreactivity in a murine model;Woods;Blood,2017

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