Design and synthesis of cyclopropane-based conformationally restricted GABA analogues as selective inhibitors for betaine/GABA transporter 1
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry
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1. Helix-forming aliphatic homo-δ-peptide foldamers based on the conformational restriction effects of cyclopropane;Organic & Biomolecular Chemistry;2023
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3. Molecular Determinants and Pharmacological Analysis for a Class of Competitive Non-transported Bicyclic Inhibitors of the Betaine/GABA Transporter BGT1;Frontiers in Chemistry;2021-09-14
4. Development, Recent Achievements and Current Directions of Research into GABA Uptake Inhibitors;Current Medicinal Chemistry;2021-03-09
5. Stereo- and regiocontrolled synthesis of highly functionalized cyclopentanes with multiple chiral centers;Synthetic Communications;2020-03-09
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