Discovery of DS42450411 as a potent orally active hepcidin production inhibitor: Design and optimization of novel 4-aminopyrimidine derivatives-Reference-Cited by-同舟云学术

Discovery of DS42450411 as a potent orally active hepcidin production inhibitor: Design and optimization of novel 4-aminopyrimidine derivatives

Published:2018-11 Issue:20 Volume:28 Page:3333-3337
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Fukuda Takeshi,Ishiyama Takashi,Katagiri Takahiro,Ueda Kenjiro^ORCID,Muramatsu Sumie,Hashimoto Masami,Aki Anri,Baba Daichi,Watanabe Kengo,Tanaka Naoki

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference8 articles.

1. Regulation of iron acquisition and storage: consequences for iron-linked disorders

2. Anemia of Chronic Disease

3. LEAP-1, a novel highly disulfide-bonded human peptide, exhibits antimicrobial activity

4. IL-6 mediates hypoferremia of inflammation by inducing the synthesis of the iron regulatory hormone hepcidin

5. Hepcidin—a regulator of intestinal iron absorption and iron recycling by macrophages

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