Discovery and optimization of aminopyrimidinones as potent and state-dependent Nav1.7 antagonists-Reference-Cited by-同舟云学术

Discovery and optimization of aminopyrimidinones as potent and state-dependent Nav1.7 antagonists

Published:2012-01 Issue:2 Volume:22 Page:1055-1060
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Nguyen Hanh Nho,Bregman Howie,Buchanan John L.,Du Bingfan,Feric Elma,Huang Liyue,Li Xingwen,Ligutti Joseph,Liu Dong,Malmberg Annika B.,Matson David J.,McDermott Jeff S.,Patel Vinod F.,Wilenkin Ben,Zou Anruo,McDonough Stefan I.,DiMauro Erin F.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference17 articles.

1. The roles of sodium channels in nociception: Implications for mechanisms of pain

2. MEXILETINE FOR TREATMENT OF CHRONIC PAINFUL DIABETIC NEUROPATHY

3. The Use of Oral Mexiletine for the Treatment of Pain after Peripheral Nerve Injury

4. A critical review of controlled clinical trials for peripheral neuropathic pain and complex regional pain syndromes

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