Design and synthesis of a novel series of [1-(4-hydroxy-benzyl)-1H-indol-5-yloxy]-acetic acid compounds as potent, selective, thyroid hormone receptor β agonists-Reference-Cited by-同舟云学术

Design and synthesis of a novel series of [1-(4-hydroxy-benzyl)-1H-indol-5-yloxy]-acetic acid compounds as potent, selective, thyroid hormone receptor β agonists

Published:2015-04 Issue:7 Volume:25 Page:1377-1380
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Burkholder Timothy P.,Cunningham Brian E.,Clayton Joshua R.,Lander Peter A.,Brown Matthew L.,Doti Robert A.,Durst Gregory L.,Montrose-Rafizadeh Chahrzad,King Constance,Osborne Harold E.,Amos Robert M.,Zink Richard W.,Stramm Lawrence E.,Burris Thomas P.,Cardona Guemalli,Konkol Debra L.,Reidy Charles,Christe Michael E.,Genin Michael J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference22 articles.

1. Selective Thyroid Hormone Receptor Modulators

2. Abnormal heart rate and body temperature in mice lacking thyroid hormone receptor alpha 1

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