Design and synthesis of potent β-secretase (BACE1) inhibitors with carboxylic acid bioisosteres-Reference-Cited by-同舟云学术

Design and synthesis of potent β-secretase (BACE1) inhibitors with carboxylic acid bioisosteres

Published:2006-05 Issue:9 Volume:16 Page:2380-2386
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Kimura Tooru,Hamada Yoshio,Stochaj Monika,Ikari Hayato,Nagamine Ayaka,Abdel-Rahman Hamdy,Igawa Naoto,Hidaka Koushi,Nguyen Jeffrey-Tri,Saito Kazuki,Hayashi Yoshio,Kiso Yoshiaki

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference32 articles.

1. Laying it on thick

2. Cellular mechanisms of beta -amyloid production and secretion

3. The molecular pathology of Alzheimer's disease

4. Structure of the Protease Domain of Memapsin 2 (β-Secretase) Complexed with Inhibitor

5. AMYLOIDOSIS

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