Design and synthesis of pyrazolo[3,4-d]pyrimidinone derivatives: Discovery of selective phosphodiesterase-5 inhibitors
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry
Reference25 articles.
1. Bruzziches R, Francomano D, Gareri P, Lenzi A, Aversa A. An update on pharmacological treatment of erectile dysfunction with phosphodiesterase type 5 inhibitors. Expert opiniononpharmacotherapy,14(10),13331344(2013),doi:10.1517/14656566.2013.799665.
2. Beavo J A. Cyclic nucleotide phosphodiesterases: functional implications of multipleisoforms.Physiologicalreviews,75,725748(1995),doi:10.1152/physrev.1995.75.4.725.
3. Isolation and characterization of PDE8A, a novel human cAMP-specific phosphodiesterase;Fisher;Biochem Biophys Res Commun,1998
4. Identification and characterization of a novel family of cyclic nucleotide phosphodiesterases;Soderling;J Biol Chem,1998
5. Thomas M K, Francis S H, Corbin J. Substrate-and kinase-directed regulation of phosphorylation of a cGMP-binding phosphodiesterase by cGMP. Journal of Biological Chemistry, 265, 14971-14978(1990), doi.org: 37232-061.
Cited by 14 articles. 订阅此论文施引文献 订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献
1. An efficient One-Pot synthesis of NaOCl mediated pyrazolopyrimidine derivatives;Results in Chemistry;2024-10
2. A novel standard‐free detection of adulteration method for sildenafil derivatives in dietary supplements;Biomedical Chromatography;2024-06-05
3. New Ciprofloxacin–Pyrazolopyrimidine Hybrids as Topoisomerase IV and Gyrase Inhibitors against MRSA AUMC 261;ChemistrySelect;2024-04-19
4. Analytical methods for the detection and characterization of unapproved phosphodiesterase type 5 inhibitors (PDE-5i) used in adulteration of dietary supplements- a review;Food Additives & Contaminants: Part A;2023-11-27
5. Novel Glu-based pyrazolo[3,4-d]pyrimidine analogues: design, synthesis and biological evaluation as DHFR and TS dual inhibitors;Journal of Enzyme Inhibition and Medicinal Chemistry;2023-04-20
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3