Design of potent thiophene inhibitors of polo-like kinase 1 with improved solubility and reduced protein binding-Reference-Cited by-同舟云学术

Design of potent thiophene inhibitors of polo-like kinase 1 with improved solubility and reduced protein binding

Published:2009-03 Issue:6 Volume:19 Page:1694-1697
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Emmitte Kyle A.,Adjebang George M.,Andrews C. Webb,Alberti Jennifer G. Badiang,Bambal Ramesh,Chamberlain Stanley D.,Davis-Ward Ronda G.,Dickson Hamilton D.,Hassler Daniel F.,Hornberger Keith R.,Jackson Jeffrey R.,Kuntz Kevin W.,Lansing Timothy J.,Mook Robert A.,Nailor Kristen E.,Pobanz Mark A.,Smith Stephon C.,Sung Chiu-Mei,Cheung Mui

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

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3. Tubulin-associated proteins: Aurora and Polo-like kinases as therapeutic targets in cancer

4. Progress in the Discovery of Polo-like Kinase Inhibitors

5. Polo-like kinases and the orchestration of cell division

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