Discovery of aryl ureas and aryl amides as potent and selective histamine H3 receptor antagonists for the treatment of obesity (Part I)-Reference-Cited by-同舟云学术

Discovery of aryl ureas and aryl amides as potent and selective histamine H3 receptor antagonists for the treatment of obesity (Part I)

Published:2013-06 Issue:11 Volume:23 Page:3416-3420
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Gao Zhongli,Hurst William J.,Guillot Etienne,Czechtizky Werngard,Lukasczyk Ulrike,Nagorny Raisa,Pruniaux Marie-Pierre,Schwink Lothar,Sanchez Juan Antonio,Stengelin Siegfried,Tang Lei,Winkler Irvin,Hendrix James A.,George Pascal G.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference29 articles.

1. Obesity: a disease or a biological adaptation? An update

2. Is severe obesity a cardiovascular health concern in the inuit population?

3. The Histamine H3 Receptor and Eating Behavior

4. Inverse Agonism and Neutral Antagonism at α1a- and α1b-Adrenergic Receptor Subtypes

5. Inverse agonism at α2-adrenoceptors in native tissue

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