Discovery of a series of novel 5H-pyrrolo[2,3-b]pyrazine-2-phenyl ethers, as potent JAK3 kinase inhibitors-Reference-Cited by-同舟云学术

Discovery of a series of novel 5H-pyrrolo[2,3-b]pyrazine-2-phenyl ethers, as potent JAK3 kinase inhibitors

Published:2013-05 Issue:9 Volume:23 Page:2522-2526
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Jaime-Figueroa Saul,De Vicente Javier,Hermann Johannes,Jahangir Alam,Jin Sue,Kuglstatter Andreas,Lynch Stephen M.,Menke John,Niu Linghao,Patel Vaishali,Shao Ada,Soth Michael,Vu Minh Diem,Yee Calvin

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference13 articles.

1. Jak and Syk: Emerging their relevance to the treatment of inflammatory diseases

2. Jaks, STATs, Cytokine Signal Transduction, and Immunoregulation: Are We There Yet?

3. Chapter 12 Advances in the Discovery of Small Molecule JAK3 Inhibitors

4. Recent patents in the discovery of small molecule inhibitors of JAK3

5. Ruxolitinib

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