Novel and potent inhibitors of stearoyl-CoA desaturase-1. Part I: Discovery of 3-(2-hydroxyethoxy)-4-methoxy-N-[5-(3-trifluoromethylbenzyl)thiazol-2-yl]benzamide-Reference-Cited by-同舟云学术

Novel and potent inhibitors of stearoyl-CoA desaturase-1. Part I: Discovery of 3-(2-hydroxyethoxy)-4-methoxy-N-[5-(3-trifluoromethylbenzyl)thiazol-2-yl]benzamide

Published:2009-08 Issue:15 Volume:19 Page:4151-4158
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Uto Yoshikazu,Ogata Tsuneaki,Harada Jun,Kiyotsuka Yohei,Ueno Yuko,Miyazawa Yuriko,Kurata Hitoshi,Deguchi Tsuneo,Watanabe Nobuaki,Takagi Toshiyuki,Wakimoto Satoko,Okuyama Ryo,Abe Manabu,Kurikawa Nobuya,Kawamura Sayako,Yamato Michiko,Osumi Jun

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. Stearoyl-CoA desaturase as a new drug target for obesity treatment

2. Recent insights into stearoyl-CoA desaturase-1

3. Identification and Characterization of Murine SCD4, a Novel Heart-specific Stearoyl-CoA Desaturase Isoform Regulated by Leptin and Dietary Factors

4. Characterization of HSCD5, a novel human stearoyl-CoA desaturase unique to primates

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