Structural basis for binding of cyclic 2-oxoglutarate analogues to factor-inhibiting hypoxia-inducible factor-Reference-Cited by-同舟云学术

Structural basis for binding of cyclic 2-oxoglutarate analogues to factor-inhibiting hypoxia-inducible factor

Published:2010-10 Issue:20 Volume:20 Page:6125-6128
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Conejo-Garcia Ana,McDonough Michael A.,Loenarz Christoph,McNeill Luke A.,Hewitson Kirsty S.,Ge Wei,Liénard Benoît M.,Schofield Christopher J.,Clifton Ian J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. Regulation of hypoxia-inducible factor 1 by prolyl and asparaginyl hydroxylases

2. The von Hippel–Lindau protein, HIF hydroxylation, and oxygen sensing

3. Signalling hypoxia by HIF hydroxylases

4. JmjC-domain-containing proteins and histone demethylation

5. The inhibition of factor inhibiting hypoxia-inducible factor (FIH) by β-oxocarboxylic acids

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