Discovery of thiadiazole amides as potent, S1P3-sparing agonists of sphingosine-1-phosphate 1 (S1P1) receptor-Reference-Cited by-同舟云学术

Discovery of thiadiazole amides as potent, S1P3-sparing agonists of sphingosine-1-phosphate 1 (S1P1) receptor

Published:2012-04 Issue:7 Volume:22 Page:2456-2459
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Xu Heng,Zhang Haibo,Luan Linbo,Xu Yan,Li Chengyong,Wang Yonghui,Han Fangbin,Yang Ting,Ren Feng,Xiang Jia-Ning,Elliott John D.,Zhao Yonggang,Guo Taylor B.,Lu Hongtao,Zhang Wei,Hirst David,Lindon Matthew,Lin Xichen

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. Fingolimod (FTY720): discovery and development of an oral drug to treat multiple sclerosis

2. FTY720: Sphingosine 1-Phosphate Receptor-1 in the Control of Lymphocyte Egress and Endothelial Barrier Function

3. FTY720 Story: Discovery of the First Sphingosine 1-Phosphate Receptor Modulator

4. Fingolimod (FTY720), the Sphingosine 1-Phosphate Receptor Modulator, as a New Therapeutic Drug in Multiple Sclerosis

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