Subtype-selective Nav1.8 sodium channel blockers: Identification of potent, orally active nicotinamide derivatives-Reference-Cited by-同舟云学术

Subtype-selective Nav1.8 sodium channel blockers: Identification of potent, orally active nicotinamide derivatives

Published:2010-11 Issue:22 Volume:20 Page:6812-6815
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Kort Michael E.,Atkinson Robert N.,Thomas James B.,Drizin Irene,Johnson Matthew S.,Secrest Matthew A.,Gregg Robert J.,Scanio Marc J.C.,Shi Lei,Hakeem Ahmed H.,Matulenko Mark A.,Chapman Mark L.,Krambis Michael J.,Liu Dong,Shieh Char-Chang,Zhang XuFeng,Simler Gricelda,Mikusa Joseph P.,Zhong Chengmin,Joshi Shailen,Honore Prisca,Roeloffs Rosemarie,Werness Stephen,Antonio Brett,Marsh Kennan C.,Faltynek Connie R.,Krafte Douglas S.,Jarvis Michael F.,Marron Brian E.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. From Ionic Currents to Molecular Mechanisms

2. Voltage-Gated Sodium Channels and Hyperalgesia

3. Voltage-Gated Sodium Channel Blockers; Target Validation and Therapeutic Potential

4. International Union of Pharmacology. XLVII. Nomenclature and Structure-Function Relationships of Voltage-Gated Sodium Channels

5. The role of voltage-gated sodium channels in neuropathic pain

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