The discovery of the potent aurora inhibitor MK-0457 (VX-680)-Reference-Cited by-同舟云学术

The discovery of the potent aurora inhibitor MK-0457 (VX-680)

Published:2009-07 Issue:13 Volume:19 Page:3586-3592
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Bebbington David,Binch Hayley,Charrier Jean-Damien,Everitt Simon,Fraysse Damien,Golec Julian,Kay David,Knegtel Ronald,Mak Chau,Mazzei Francesca,Miller Andrew,Mortimore Michael,O’Donnell Michael,Patel Sanjay,Pierard Francoise,Pinder Joanne,Pollard John,Ramaya Sharn,Robinson Daniel,Rutherford Alistair,Studley John,Westcott James

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference31 articles.

1. Mutations in aurora prevent centrosome separation leading to the formation of monopolar spindles

2. Aurora Kinases as Anticancer Drug Targets

3. Aurora-kinase inhibitors as anticancer agents

4. Aurora kinases: shining lights on the therapeutic horizon?

Cited by 91 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Novel sulfonamide-indolinone hybrids targeting mitochondrial respiration of breast cancer cells;European Journal of Medicinal Chemistry;2024-03

2. Global Reactivity Profiling of the Catalytic Lysine in Human Kinome for Covalent Inhibitor Development;Angewandte Chemie;2024-02-14

3. Global Reactivity Profiling of the Catalytic Lysine in Human Kinome for Covalent Inhibitor Development;Angewandte Chemie International Edition;2024-02-14

4. Recent Synthetic and Biological Developments on 1,2,4‐Triazolopyrimidines;ChemistrySelect;2023-09-04

5. The Importance of the Pyrazole Scaffold in the Design of Protein Kinases Inhibitors as Targeted Anticancer Therapies;Molecules;2023-07-12