Total synthesis and evaluation of 22-(3-azidobenzoyloxy)methyl epothilone C for photoaffinity labeling of β-tubulin-Reference-Cited by-同舟云学术

Total synthesis and evaluation of 22-(3-azidobenzoyloxy)methyl epothilone C for photoaffinity labeling of β-tubulin

Published:2009-06 Issue:12 Volume:19 Page:3293-3296
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Hutt Oliver E.,Inagaki Jun,Reddy Bollu S.,Nair Sajiv K.,Reiff Emily A.,Henri John T.,Greiner Jack F.,VanderVelde David G.,Chiu Ting-Lan,Amin Elizabeth A.,Himes Richard H.,Georg Gunda I.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference24 articles.

1. Epothilons A and B: Antifungal and Cytotoxic Compounds from Sorangium cellulosum (Myxobacteria). Production, Physico-chemical and Biological Properties.

2. Understanding tubulin-Taxol interactions: Mutations that impart Taxol binding to yeast tubulin

3. A Unified and Quantitative Receptor Model for the Microtubule Binding of Paclitaxel and Epothilone

4. A common pharmacophore for cytotoxic natural products that stabilize microtubules

5. A Common Pharmacophore for Taxol and the Epothilones Based on the Biological Activity of a Taxane Molecule Lacking a C-13 Side Chain

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1. Characterizing the Epothilone Binding Site on β-Tubulin by Photoaffinity Labeling: Identification of β-Tubulin Peptides TARGSQQY and TSRGSQQY as Targets of an Epothilone Photoprobe for Polymerized Tubulin;Journal of Medicinal Chemistry;2016-03-17

2. Selected hybrid natural products as tubulin modulators;European Journal of Medicinal Chemistry;2015-04

3. Epothilones: From Discovery to Clinical Trials;Current Topics in Medicinal Chemistry;2014-12-12

4. Epothilones as Lead Structures for New Anticancer Drugs;Drug Discovery from Natural Products;2012-09-13

5. Chapter 16. Epothilones as Lead Structures for New Anticancer Drugs;Drug Discovery;2012