Syntheses and biological evaluation of 5-(piperidin-1-yl)-3-phenyl-pentylsulfones as CCR5 antagonists-Reference-Cited by-同舟云学术

Syntheses and biological evaluation of 5-(piperidin-1-yl)-3-phenyl-pentylsulfones as CCR5 antagonists

Published:2004-07 Issue:13 Volume:14 Page:3589-3593
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Shankaran K.,Donnelly Karla L.,Shah Shrenik K.,Caldwell Charles G.,Chen Ping,Finke Paul E.,Oates Bryan,MacCoss Malcolm,Mills Sander G.,DeMartino Julie A.,Gould Sandra L.,Malkowitz Lorraine,Siciliano Salvatore J.,Springer Martin S.,Kwei Gloria,Carella Anthony,Carver Gwen,Danzeisen Renee,Hazuda Daria,Holmes Karen,Kessler Joseph,Lineberger Janet,Miller Michael D.,Emini Emilio A.,Schleif William A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference31 articles.

1. Chemokine Receptors and Chemokines in HIV Infection

2. Chemokine Receptors As HIV Co-Receptors: Targets for Therapeutic Intervention in AIDS

3. Opportunities for novel therapeutic agents acting at chemokine receptors

4. Recent developments in modulating chemokine networks

5. Identification of RANTES, MIP-1α, and MIP-1β as the Major HIV-Suppressive Factors Produced by CD8 + T Cells

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