Discovery of bisamide-heterocycles as inhibitors of scavenger receptor BI (SR-BI)-mediated lipid uptake-Reference-Cited by-同舟云学术

Discovery of bisamide-heterocycles as inhibitors of scavenger receptor BI (SR-BI)-mediated lipid uptake

Published:2015-06 Issue:12 Volume:25 Page:2594-2598
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Dockendorff Chris,Faloon Patrick W.,Germain Andrew,Yu Miao,Youngsaye Willmen,Nag Partha P.,Bennion Melissa,Penman Marsha,Nieland Thomas J.F.,Dandapani Sivaraman,Perez José R.,Munoz Benito,Palmer Michelle A.,Schreiber Stuart L.,Krieger Monty

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference33 articles.

1. Identification of Scavenger Receptor SR-BI as a High Density Lipoprotein Receptor

2. The Role of the High-Density Lipoprotein Receptor SR-BI in the Lipid Metabolism of Endocrine and Other Tissues

3. Exoplasmic cysteine Cys384 of the HDL receptor SR-BI is critical for its sensitivity to a small-molecule inhibitor and normal lipid transport activity

4. Extracellular Disulfide Bonds Support Scavenger Receptor Class B Type I-Mediated Cholesterol Transport

5. Glycine Dimerization Motif in the N-terminal Transmembrane Domain of the High Density Lipoprotein Receptor SR-BI Required for Normal Receptor Oligomerization and Lipid Transport

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3. Inhibition of Scavenger Receptor Class B Type 1 (SR-B1) Expression and Activity as a Potential Novel Target to Disrupt Cholesterol Availability in Castration-Resistant Prostate Cancer;Pharmaceutics;2021-09-18

4. Cholesterol uptake and efflux are impaired in human trophoblast cells from pregnancies with maternal supraphysiological hypercholesterolemia;Scientific Reports;2020-03-24

5. Metal‐Free Synthesis of Methylene‐Bridged Bisamide via Selectfluor‐Mediated Oxidative Methylenation;ChemistrySelect;2018-12-07