Design, synthesis and biological evaluation of substituted 3-amino-N-(thiazol-2-yl)pyrazine-2-carboxamides as inhibitors of mycobacterial methionine aminopeptidase 1-Reference-Cited by-同舟云学术

Design, synthesis and biological evaluation of substituted 3-amino-N-(thiazol-2-yl)pyrazine-2-carboxamides as inhibitors of mycobacterial methionine aminopeptidase 1

Published:2022-01 Issue: Volume:118 Page:105489
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Juhás Martin,Pallabothula Vinod S.K.,Grabrijan Katarina,Šimovičová Martina,Janďourek Ondřej,Konečná Klára,Bárta Pavel,Paterová Pavla,Gobec Stanislav,Sosič Izidor,Zitko Jan

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference52 articles.

1. Geneva: World Health Organization, Global Tuberculosis Report 2020, 2020.

2. Nontuberculous mycobacterial pulmonary infections;Johnson;J. Thorac. Dis.,2014

3. Characteristics of Nontuberculous Mycobacterial Infections at a Midwestern Tertiary Hospital: A Retrospective Study of 365 Patients;Hannah;Open Forum Infectious Diseases,2020

4. Mycobacterial outer membrane is a lipid bilayer and the inner membrane is unusually rich in diacyl phosphatidylinositol dimannosides;Bansal-Mutalik;Proc. Natl. Acad. Sci. U.S.A.,2014

5. The tuberculous granuloma: an unsuccessful host defence mechanism providing a safety shelter for the bacteria?;Silva Miranda;Clin. Dev. Immunol.,2012

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