A combine approach of chemical synthesis, biological evaluation and structural dynamics studies revealed thiazole substituted arylamine derivatives as potent FabH enzyme inhibitors-Reference-Cited by-同舟云学术

A combine approach of chemical synthesis, biological evaluation and structural dynamics studies revealed thiazole substituted arylamine derivatives as potent FabH enzyme inhibitors

Published:2020-12 Issue: Volume:105 Page:104426
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Ahmad Haseen,Ahmad Faisal,Parveen Shaista,Ahmad Sajjad,Azam Syed Sikander,Hassan Abbas

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference60 articles.

1. The evolution of antibiotic resistance;MacLean;Science (80-),2019

2. Global priority list of antibiotic-resistant bacteria to guide research, discovery, and development of new antibiotics;Tacconelli;World Heal. Organ,2017

3. Computer-aided drug design methods;Yu,2017

4. R.J. Heath, C.O. Rock, Fatty acid biosynthesis as a target for novel antibacterials, Curr. Opin. Investig. Drugs (London, Engl. 2000). 5 (2004) 146.

5. Bacterial fatty acid biosynthesis: targets for antibacterial drug discovery;Campbell;Annu. Rev. Microbiol.,2001

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